bit [ASAP] Design, Synthesis, and Pharmacological Evaluation of Second Generation EZH2 Inhibitors with Long Residence Time By feedproxy.google.com Published On :: Thu, 02 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00045 Full Article
bit [ASAP] Structure Optimization of Gatastatin for the Development of ?-Tubulin-Specific Inhibitor By feedproxy.google.com Published On :: Mon, 06 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00526 Full Article
bit [ASAP] Chiral Analogues of PFI-1 as BET Inhibitors and Their Functional Role in Myeloid Malignancies By feedproxy.google.com Published On :: Tue, 07 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00625 Full Article
bit [ASAP] Rationally Designed Covalent BCL6 Inhibitor That Targets a Tyrosine Residue in the Homodimer Interface By feedproxy.google.com Published On :: Tue, 07 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00111 Full Article
bit [ASAP] Exploring the Implication of DDX3X in DENV Infection: Discovery of the First-in-Class DDX3X Fluorescent Inhibitor By feedproxy.google.com Published On :: Thu, 09 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00681 Full Article
bit [ASAP] Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction By feedproxy.google.com Published On :: Fri, 10 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00594 Full Article
bit [ASAP] New Dual CK2/HDAC1 Inhibitors with Nanomolar Inhibitory Activity against Both Enzymes By feedproxy.google.com Published On :: Fri, 10 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00561 Full Article
bit [ASAP] Design and Synthesis of Tetrazole- and Pyridine-Containing Itraconazole Analogs as Potent Angiogenesis Inhibitors By feedproxy.google.com Published On :: Mon, 13 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.9b00438 Full Article
bit [ASAP] Artemisinin Derivatives with Antimelanoma Activity Show Inhibitory Effect against Human DNA Topoisomerase 1 By feedproxy.google.com Published On :: Tue, 14 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00131 Full Article
bit [ASAP] Discovery of a Potent Dual Inhibitor of Wild-Type and Mutant Respiratory Syncytial Virus Fusion Proteins By feedproxy.google.com Published On :: Wed, 15 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00008 Full Article
bit [ASAP] Characterization of Specific <italic toggle="yes">N</italic>-a-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library By feedproxy.google.com Published On :: Wed, 15 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00029 Full Article
bit [ASAP] Discovery of an Atropisomeric PI3Kß Selective Inhibitor through Optimization of the Hinge Binding Motif By feedproxy.google.com Published On :: Wed, 15 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00095 Full Article
bit [ASAP] Discovery of CPI-1612: A Potent, Selective, and Orally Bioavailable EP300/CBP Histone Acetyltransferase Inhibitor By feedproxy.google.com Published On :: Mon, 27 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00155 Full Article
bit [ASAP] Development of Selective Steroid Inhibitors for the Glucose-6-phosphate Dehydrogenase from <italic toggle="yes">Trypanosoma cruzi</italic> By feedproxy.google.com Published On :: Wed, 29 Apr 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00106 Full Article
bit [ASAP] Discovery of Adamantane Carboxamides as Ebola Virus Cell Entry and Glycoprotein Inhibitors By feedproxy.google.com Published On :: Fri, 01 May 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00025 Full Article
bit [ASAP] Benzoxazepine-Derived Selective, Orally Bioavailable Inhibitor of Human Acidic Mammalian Chitinase By feedproxy.google.com Published On :: Fri, 01 May 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00092 Full Article
bit [ASAP] Scaffold Repurposing of in-House Chemical Library toward the Identification of New Casein Kinase 1 d Inhibitors By feedproxy.google.com Published On :: Mon, 04 May 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00028 Full Article
bit [ASAP] Synthesis and Evaluation of <sup>11</sup>C- and <sup>18</sup>F-Labeled SOAT1 Inhibitors as Macrophage Foam Cell Imaging Agents By feedproxy.google.com Published On :: Wed, 06 May 2020 04:00:00 GMT ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.0c00127 Full Article
bit Djordje Ozbolt: regaining memory loss / exhibition curator, Nicoletta Lambertucci By library.mit.edu Published On :: Sun, 23 Feb 2020 06:00:02 EST Rotch Library - N6488.I8 V433 2019 Y8 Full Article
bit T.C. Cannon: at the edge of America / edited by Karen Kramer ; with contributions by heather ahtone, Sherwin Bitsui, Caitlin Cooper, Frank Buffalo Hyde, Trevor Fairbrother, Santee Frazier, Joy Harjo, Joan Naviyuk Kane, Karen Kramer, Deana McCloud, America By library.mit.edu Published On :: Sun, 23 Feb 2020 06:00:02 EST Rotch Library - NX512.C36 A4 2018 Full Article
bit Ghana freedom: Ghana pavilion at the 58th International Art Exhibition La Biennale di Venezia By library.mit.edu Published On :: Sun, 23 Feb 2020 06:00:02 EST Rotch Library - N6488.I8 V433 2019 G4 Full Article
bit My art guide: Venice 2019, 58th Biennale Arte: national participations, collateral events, exhibitions, events, museums, foundations, restaurants, hotels, city maps By library.mit.edu Published On :: Sun, 23 Feb 2020 06:00:02 EST Rotch Library - N6488.I8 V433 2019 A11 Full Article
bit Democracy and imperialism: Irving Babbitt and warlike democracies / William S. Smith By library.mit.edu Published On :: Sun, 2 Feb 2020 08:57:26 EST Dewey Library - JZ1480.S5446 2019 Full Article
bit Mr Dog and the rabbit habit / Ben Fogle ; with Steve Cole ; [illustrations by Nikolas Ilic] By darius.uleth.ca Published On :: Fogle, Ben, 1973- author Full Article
bit Beyond temperature: controlling collagen fibrillogenesis under physiological conditions via interaction with cucurbit[7]uril By feeds.rsc.org Published On :: Chem. Commun., 2020, 56,4946-4949DOI: 10.1039/D0CC01444C, CommunicationQiuping Xie, Delong Hou, Jinming Chang, Zhou Xu, Qi Zeng, Zhonghui Wang, Yi ChenA supramolecular strategy as efficient as temperature that enabled facile control over collagen fibrillogenesis under physiological conditions was reported.The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
bit Discovery of [1,2,4]triazolo[4,3-a]pyrazine derivatives bearing 4-oxo-pyridazinone moiety as potential c-Met kinase inhibitors By feeds.rsc.org Published On :: New J. Chem., 2020, Accepted ManuscriptDOI: 10.1039/D0NJ00575D, PaperBinliang Zhang, Xiaobo Liu, Hehua Xiong, Qian Zhang, Xin Sun, Zunhua Yang, Shan Xu, Pengwu Zheng, Wufu ZhuTwo series of [1,2,4]triazolo[4,3-a]pyrazine derivatives bearing 4-oxo-pyridazinone moiety (compounds 21a-l and 22a-l) were designed and evaluated for the IC50 values against three cancer cell lines (A549, MCF-7 and Hela) and...The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
bit Whole Genome Sequence Analysis and Homology Modelling of Main Protease and Non-Structural Protein 3 of the SARS-CoV-2 reveals an Aza-Peptide and a Lead Inhibitor with Possible Antiviral Properties By feeds.rsc.org Published On :: New J. Chem., 2020, Accepted ManuscriptDOI: 10.1039/D0NJ00974A, PaperArun K Shankar, Divya Bhanu, Anjani Alluri, Samriddhi GuptaThe family of viruses belonging to Coronaviridae consist of virulent pathogens that have a zoonotic property, Severe Acute Respiratory Syndrome (SARS-CoV) and Middle East Respiratory Syndrome (MERS-CoV) of this family...The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
bit POM-based dyes featured rigidified bithiophene π linkers: Potential high-efficient dyes for dye-sensitized solar cells By feeds.rsc.org Published On :: New J. Chem., 2020, Accepted ManuscriptDOI: 10.1039/D0NJ01150A, PaperYu Gao, Li-Kai Yan, Wei Guan, Yanhong XuA series of POM-based dyes with triphenylamine electron donor group, cyanoacrylic acid electron acceptor group and different π linkers of thiophene derivatives are systematically investigated to analyze the influence of...The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
bit [ASAP] Structural and Biological Basis of Small Molecule Inhibition of <italic toggle="yes">Escherichia coli</italic> LpxD Acyltransferase Essential for Lipopolysaccharide Biosynthesis By dx.doi.org Published On :: Thu, 22 Aug 2019 04:00:00 GMT ACS Infectious DiseasesDOI: 10.1021/acsinfecdis.9b00127 Full Article
bit [ASAP] Broad Spectrum ß-Lactamase Inhibition by a Thioether Substituted Bicyclic Boronate By dx.doi.org Published On :: Mon, 06 Jan 2020 05:00:00 GMT ACS Infectious DiseasesDOI: 10.1021/acsinfecdis.9b00330 Full Article
bit [ASAP] Advancement of GyrB Inhibitors for Treatment of Infections Caused by <italic toggle="yes">Mycobacterium tuberculosis</italic> and Non-tuberculous Mycobacteria By dx.doi.org Published On :: Wed, 25 Mar 2020 04:00:00 GMT ACS Infectious DiseasesDOI: 10.1021/acsinfecdis.0c00025 Full Article
bit [ASAP] Small Molecule Carboxylates Inhibit Metallo-ß-lactamases and Resensitize Carbapenem-Resistant Bacteria to Meropenem By dx.doi.org Published On :: Fri, 03 Apr 2020 04:00:00 GMT ACS Infectious DiseasesDOI: 10.1021/acsinfecdis.9b00459 Full Article
bit Now on View–“Padlocked”: New York’s Prohibition Years By blog.nyhistory.org Published On :: Wed, 06 Mar 2019 15:00:19 +0000 Set to commence on January 17, 1920, the great social experiment of Prohibition had already begun with a “dry run” for Americans adapting to the restriction of alcohol inspired by World War I. That was followed by a full year anticipating the event through the process of Constitutional amendment and the passage of enforcement legislation... The post Now on View–“Padlocked”: New York’s Prohibition Years appeared first on New-York Historical Society. Full Article Ephemera Exhibitions 18th amendment 21st amendment Alcohol bootleggers flappers now on view Prohibition repeal speakeasy Stork Club Temperance Volstead Act
bit United Nations protection of humanity and its habitat : a new international law of security and protection / by Bertrand G. Ramcharan By prospero.murdoch.edu.au Published On :: Ramcharan, B. G., author Full Article
bit Inside the Equal Access to Justice Act : environmental litigation and the crippling battle over America's lands, endangered species, and critical habitats / Lowell E. Baier By prospero.murdoch.edu.au Published On :: Baier, Lowell E., author Full Article
bit The habitats directive in its EU environmental law context : European nature's best hope? / edited by Charles-Hubert Born, An Cliquet, Hendrik Schoukens, Delphine Misonne, and Geert Van Hoorick By prospero.murdoch.edu.au Published On :: Full Article
bit Humanitarian intervention as an exception to the prohibition on the use of force / Petra Zvržina By prospero.murdoch.edu.au Published On :: Zvržina, Petra, author Full Article
bit Social Services Legislation Amendment (Cashless Debit Card Trial Expansion) Bill 2018 [Provisions] / The Senate, Community Affairs Legislation Committee By prospero.murdoch.edu.au Published On :: Australia. Parliament. Senate. Community Affairs Legislation Committee, author, issuing body Full Article
bit The UNCITRAL model law after twenty-five years : global perspectives on international commercial arbitration / Frédéric Bachand, Fabien Gélinas, edtors By prospero.murdoch.edu.au Published On :: Full Article
bit Handbook of ICC arbitration : commentary, precedents, materials / Thomas H. Webster, Michael Buhler By prospero.murdoch.edu.au Published On :: Webster, Thomas H, author Full Article
bit A guide to the UNCITRAL Model Law on International Commercial Arbitration : legislative history and commentary / by Howard M. Holtzmann and Joseph E. Neuhaus By prospero.murdoch.edu.au Published On :: Holtzmann, Howard M Full Article
bit Law and practice of arbitration and conciliation By prospero.murdoch.edu.au Published On :: Malhotra, O. P. (Om Prakash), 1923- author Full Article
bit Counsel as client's first enemy in arbitration? / Ugo Draetta By prospero.murdoch.edu.au Published On :: Draetta, Ugo, author Full Article
bit Collection of procedural decisions in ICC arbitration 1993-1996 = Recueil des décisions de procédure dans l'arbitrage CCI / Dominique Hascher By prospero.murdoch.edu.au Published On :: Hascher, Dominique Full Article
bit Galilee Basin (Coal Prohibition) Bill 2018 / The Senate Environment and Communications Legislation Committe By prospero.murdoch.edu.au Published On :: Australia. Parliament. Senate. Environment and Communications Legislation Committee, author, issuing body Full Article
bit The leading arbitrators' guide to international arbitration / editors, Lawrence W. Newman, Richard D. Hill By prospero.murdoch.edu.au Published On :: Full Article
bit Social Security (Administration) Amendment (Income Management to Cashless Debit Card Transition) Bill 2019 [Provisions] / The Senate, Community Affairs Legislation Committee By prospero.murdoch.edu.au Published On :: Australia. Parliament. Senate. Community Affairs Legislation Committee, author, issuing body Full Article
bit Treasury Laws Amendment (Prohibiting Energy Market Misconduct) Bill 2019 [Provisions] / Economics Legislation Committee By prospero.murdoch.edu.au Published On :: Australia. Parliament. Senate. Economics Legislation Committee, author, issuing body Full Article
bit The Bitter History of Elections By podcast.history.org Published On :: Mon, 05 Nov 2012 13:00:12 +0000 Political parties were new, the losers became Vice Presidents, and negative campaigning was finding its feet in the election of 1796. Professor Jack Lynch has the history. Full Article Government election voting
bit A three-in-one crystal of mixed sized cucurbit[n]uril homologues By feeds.rsc.org Published On :: CrystEngComm, 2020, 22,2900-2903DOI: 10.1039/D0CE00296H, CommunicationOksana Danylyuk, Volodymyr SashukCrystallization-driven self-assembly of three macrocyclic members of the cucurbit[n]uril family is explained by the cumulative effect of multiple C–H⋯O hydrogen bonds.The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
