sap [ASAP] Crystallization-Induced Diastereoisomer Transformation of Dihydroartemisinic Aldehyde with the Betti Base By feedproxy.google.com Published On :: Tue, 14 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00481 Full Article
sap [ASAP] Continuous Flow Photo-oxidations Using Supported Photocatalysts on Silica By feedproxy.google.com Published On :: Thu, 16 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00420 Full Article
sap [ASAP] Straightforward Access to 2-Iodoindolizines via Iodine-Mediated Cyclization of 2-Pyridylallenes By feedproxy.google.com Published On :: Thu, 16 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00418 Full Article
sap [ASAP] Comparing Gas–Liquid Segmented and Tube-in-Tube Setups for the Aerobic Dimerization of Desmethoxycarpacine with an Automated Flow Platform By feedproxy.google.com Published On :: Wed, 22 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00525 Full Article
sap [ASAP] A Perspective on Continuous Flow Chemistry in the Pharmaceutical Industry By feedproxy.google.com Published On :: Thu, 23 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00524 Full Article
sap [ASAP] Evaluation of Sponge Metal Catalysts in a Trickle Bed Reactor for the Continuous Hydrogenation of an Aliphatic Nitro Intermediate By feedproxy.google.com Published On :: Fri, 24 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00447 Full Article
sap [ASAP] Copper(I) Diphosphine Bifluoride Complexes as Efficient Preactivated Catalysts for Nucleophilic Addition on Unsaturated Functional Groups By feedproxy.google.com Published On :: Fri, 24 Jan 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00443 Full Article
sap [ASAP] Development of a Robust Protocol for the Synthesis of 6-Hydroxybenzofuran-3-carboxylic Acid By feedproxy.google.com Published On :: Mon, 03 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00546 Full Article
sap [ASAP] Development of a General Automated Flow Photoredox <sup>18</sup>F-Difluoromethylation of N-Heteroaromatics in an AllinOne Synthesizer By feedproxy.google.com Published On :: Thu, 06 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00442 Full Article
sap [ASAP] From Industrial Method to the Use of Silylated P(III) Reagents for the Synthesis of Relevant Phosphonylated Molecules By feedproxy.google.com Published On :: Thu, 06 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00490 Full Article
sap [ASAP] Carbon as a Simple Support for Redox Biocatalysis in Continuous Flow By feedproxy.google.com Published On :: Tue, 11 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00410 Full Article
sap [ASAP] Recent Progress in Continuous Crystallization of Pharmaceutical Products: Precise Preparation and Control By feedproxy.google.com Published On :: Thu, 13 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00362 Full Article
sap [ASAP] Total Synthesis of (+)-Oxo-tomaymycin By feedproxy.google.com Published On :: Mon, 17 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00009 Full Article
sap [ASAP] Straightforward Access to a Great Diversity of Complex Biorelevant ?-Lactams Thanks to a Tunable Cascade Multicomponent Process By feedproxy.google.com Published On :: Thu, 20 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00438 Full Article
sap [ASAP] Synthesis of 5-Substituted 1<italic toggle="yes">H</italic>-Tetrazoles from Nitriles by Continuous Flow: Application to the Synthesis of Valsartan By feedproxy.google.com Published On :: Fri, 21 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00526 Full Article
sap [ASAP] Exploring Homogeneous Conditions for Mild Buchwald–Hartwig Amination in Batch and Flow By feedproxy.google.com Published On :: Mon, 24 Feb 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00018 Full Article
sap [ASAP] What Elements Contribute to a High-Quality Continuous Processing Submission for <italic toggle="yes">OPR&D</italic>? By feedproxy.google.com Published On :: Fri, 06 Mar 2020 05:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00020 Full Article
sap [ASAP] Scalable Aerobic Oxidation of Alcohols Using Catalytic DDQ/HNO<sub>3</sub> By feedproxy.google.com Published On :: Wed, 18 Mar 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00513 Full Article
sap [ASAP] Continuous Flow Conditions for High Temperature Formation of a Benzodioxan Pharmaceutical Intermediate: Rapid Scaleup for Early Phase Material Delivery By feedproxy.google.com Published On :: Tue, 31 Mar 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00499 Full Article
sap [ASAP] An Economical Route to Lamivudine Featuring a Novel Strategy for Stereospecific Assembly By feedproxy.google.com Published On :: Fri, 10 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00083 Full Article
sap [ASAP] Playing with Fire? A Safe and Effective Deactivation of Raney Cobalt using Aqueous Sodium Nitrate By feedproxy.google.com Published On :: Mon, 13 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00053 Full Article
sap [ASAP] Nontraditional Application of the Photo-Fenton Process: A Novel Strategy for Molecular Construction Using Formamide and Flow Chemistry By feedproxy.google.com Published On :: Mon, 13 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00057 Full Article
sap [ASAP] Development of an Efficient Synthetic Process for Broflanilide By feedproxy.google.com Published On :: Wed, 15 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00028 Full Article
sap [ASAP] Green Chemistry Articles of Interest to the Pharmaceutical Industry By feedproxy.google.com Published On :: Thu, 16 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00154 Full Article
sap [ASAP] Reductive Amination Bicarbonate Quench: Gas-Evolving Waste Stream Near-Miss Investigation By feedproxy.google.com Published On :: Thu, 16 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00085 Full Article
sap [ASAP] Safety Case Study. Intrinsic Instability of Concentrated Solutions of Alcoholic Hydrogen Chloride: Potential Hazards Associated with Methanol By feedproxy.google.com Published On :: Fri, 17 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00034 Full Article
sap [ASAP] Development of a Robust and Highly Selective Ru(II)-Catalyzed Dynamic Kinetic Resolution Used to Manufacture AMG 232 By feedproxy.google.com Published On :: Fri, 17 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00427 Full Article
sap [ASAP] Scalable Synthesis of Esp and Rhodium(II) Carboxylates from Acetylacetone and RhCl<sub>3</sub>·<italic toggle="yes">x</italic>H<sub>2</sub>O By feedproxy.google.com Published On :: Tue, 21 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00164 Full Article
sap [ASAP] Investigating Process Variables and Additive Selection To Optimize Polymorphic Control of Carbamazepine in a CO<sub>2</sub> Antisolvent Crystallization Process By feedproxy.google.com Published On :: Wed, 22 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00545 Full Article
sap [ASAP] Photo-oxidation of Cyclopentadiene Using Continuous Processing: Application to the Synthesis of (1<italic toggle="yes">R</italic>,4<italic toggle="yes">S</italic>)-4-Hydroxycyclopent-2-en-1-yl Acetate By feedproxy.google.com Published On :: Wed, 22 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00066 Full Article
sap [ASAP] Update to Our Reader, Reviewer, and Author Communities—April 2020 By feedproxy.google.com Published On :: Thu, 23 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00194 Full Article
sap [ASAP] Efficient Kinetic Data Acquisition and Model Prediction: Continuous Flow Microreactors, Inline Fourier Transform Infrared Spectroscopy, and Self-Modeling Curve Resolution By feedproxy.google.com Published On :: Mon, 27 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00037 Full Article
sap [ASAP] Process Development and Large-Scale Synthesis of BTK Inhibitor BIIB068 By feedproxy.google.com Published On :: Mon, 27 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00087 Full Article
sap [ASAP] A Versatile Electrochemical Batch Reactor for Synthetic Organic and Inorganic Transformations and Analytical Electrochemistry By feedproxy.google.com Published On :: Mon, 27 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00091 Full Article
sap [ASAP] Improved Synthesis of 6-Chloro-5-methylpyridin-2-amine: A Key Intermediate for Making Lumacaftor By feedproxy.google.com Published On :: Tue, 28 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00556 Full Article
sap [ASAP] <italic toggle="yes">N</italic>-Acyl-5,5-Dimethylhydantoins: Mild Acyl-Transfer Reagents for the Synthesis of Ketones Using Pd–PEPPSI or Pd/Phosphine Catalysts By feedproxy.google.com Published On :: Tue, 28 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00054 Full Article
sap [ASAP] Drug Loading and Dissolution Properties of Dalcetrapib–Montmorillonite Nanocomposite Microparticles By feedproxy.google.com Published On :: Wed, 29 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00460 Full Article
sap [ASAP] Bromine–Lithium Exchange on a <italic toggle="yes">gem</italic>-Dibromoalkene, Part 2: Comparative Performance of Flow Micromixers By feedproxy.google.com Published On :: Thu, 30 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00203 Full Article
sap [ASAP] A Scalable Membrane Pervaporation Approach for Continuous Flow Olefin Metathesis By feedproxy.google.com Published On :: Thu, 30 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00061 Full Article
sap [ASAP] Scalable Synthesis of <italic toggle="yes">S</italic>-Fluoromethyl Benzenesulfonothioate By feedproxy.google.com Published On :: Thu, 30 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00101 Full Article
sap [ASAP] Upscaling Photoredox Cross-Coupling Reactions in Batch Using Immersion-Well Reactors By feedproxy.google.com Published On :: Thu, 30 Apr 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00070 Full Article
sap [ASAP] Optimized Synthesis of 7-Azaindazole by a Diels–Alder Cascade and Associated Process Safety By feedproxy.google.com Published On :: Fri, 01 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00184 Full Article
sap [ASAP] Enzymatic Preparation of the Chiral (<italic toggle="yes">S</italic>)-Sulfoxide Drug Esomeprazole at Pilot-Scale Levels By feedproxy.google.com Published On :: Sun, 03 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00115 Full Article
sap [ASAP] Continuous Process for Preparing the Difluoromethylating Reagent [(DMPU)<sub>2</sub>Zn(CF<sub>2</sub>H)<sub>2</sub>] and Improved Synthesis of the ICHF<sub>2</sub> Precursor By feedproxy.google.com Published On :: Tue, 05 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00089 Full Article
sap [ASAP] Development and Production of an Enantioselective Tetrahydroisoquinoline Synthesis Enabled by Continuous Cryogenic Lithium–Halogen Exchange By feedproxy.google.com Published On :: Tue, 05 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00141 Full Article
sap [ASAP] Some Items of Interest to Process R&D Chemists and Engineers By feedproxy.google.com Published On :: Tue, 05 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00197 Full Article
sap [ASAP] <sc>d</sc>-Serine as a Key Building Block: Enzymatic Process Development and Smart Applications within the Cascade Enzymatic Concept By feedproxy.google.com Published On :: Thu, 07 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00024 Full Article
sap [ASAP] Correction to “Application of Crabtree/Pfaltz-type Iridium Complexes for the Catalyzed Asymmetric Hydrogenation of an Agrochemical Building Block” By feedproxy.google.com Published On :: Fri, 08 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.0c00206 Full Article
sap [ASAP] Catalyst-Free Cyclization- and Curtius Rearrangement-Induced Functional Group Transformation: An Improved Synthetic Strategy of First-in-Class ATX Inhibitor Ziritaxestat (GLPG-1690) By feedproxy.google.com Published On :: Fri, 08 May 2020 04:00:00 GMT Organic Process Research & DevelopmentDOI: 10.1021/acs.oprd.9b00511 Full Article
sap The effect of crystallite size on low-temperature hydrothermal stability of Cu-SAPO-34 By feeds.rsc.org Published On :: Catal. Sci. Technol., 2020, Advance ArticleDOI: 10.1039/D0CY00414F, PaperJinpeng Du, Xiaoyan Shi, Yulong Shan, Yingjie Wang, Wenshuo Zhang, Yunbo Yu, Wenpo Shan, Hong HeTwo Cu-SAPO-34 catalysts with different crystallite sizes were obtained, and catalyst with smaller crystallite size had better low-temperature hydrothermal stability because of less Cu2+ species on the surface.To cite this article before page numbers are assigned, use the DOI form of citation above.The content of this RSS Feed (c) The Royal Society of Chemistry Full Article
